Agents
Phenothiazines
- Chlorpromazine (Largactil, Thorazine) (see Chlorpromazine, [[Chlorpromazine]])
- Prochlorperazine (Compazine) (see Prochlorperazine, [[Prochlorperazine]])
- Promethazine (Phenergan) (see Promethazine, [[Promethazine]]): phenothiazine derivative
Butryophenones
- Droperidol (Inapsine, Droleptan, Dridol, Xomolix, Innovar) (see Droperidol, [[Droperidol]])
- Haloperidol (Haldol) (see Haloperidol, [[Haloperidol]])
Benzamides
- Domperidone (Motilium) (see Domperidone, [[Domperidone]])
- Metoclopramide (Reglan) (see Metoclopramide, [[Metoclopramide]])
- Low Dose: central and peripheral dopamine D2 receptor antagonism
- High Dose: weak 5HT3 antagonism
- Enhances acetylcholine release and stimulates cholinergic receptors on gastric smooth muscle
- Trimethobenzamide
Atypical Anti-Psychotics (Also Exhibit Serotonergic Antagonism)
- Clozapine (Clozaril) (see Clozapine, [[Clozapine]])
- Olanzapine (Zyprexa) (see Olanzapine, [[Olanzapine]])
- Quetiapine (Seroquel) (see Quetiapine, [[Quetiapine]])
- Risperidone (Risperdal) (see Risperidone, [[Risperidone]])
- Ziprasidone (Geodon) (see Ziprasidone, [[Ziprasidone]])
Tricyclic Antidepressants
- Amoxapine (see Amoxapine, [[Amoxapine]])
- Clomipramine (see Clomipramine, [[Clomipramine]])
- Trimipramine (see Trimipramine, [[Trimipramine]])
Contraindications
- Parkinson’s Disease (see Parkinson’s Disease, [[Parkinsons Disease]])
References
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