α-Adrenergic Receptor Antagonists
Agents
Non-Selective α-Adrenergic Receptor Antagonists
- Phenoxybenzamine (see Phenoxybenzamine)
- Phentolamine (Regitine) (see Phentolamine)
- Tolazoline
- Trazodone (see Trazodone)
- Typical and Atypical Antipsychotics
- Olanzapine (Zyprexa) (see Olanzapine)
- Potent Serotonin 5-HT2A and 5-HT2C, Dopamine D1-4, Histamine H1, and α1-Adrenergic Receptor Antagonism
- Moderate Serotonin 5-HT3 and Muscarinic M1-5 Receptor Antagonism
- Weak Binding to GABA-A, BZD, and β-Adrenergic Receptors
- Quetiapine (Seroquel) (see Quetiapine)
- Brain Serotonin 5-HT1A and 5-HT2, Dopamine D1 and D2, Histamine H1, and α1 and α2 Adrenergic Receptor Antagonism
- Risperidone (Risperdal) (see Risperidone)
- Potent Serotonin 5-HT2, Dopamine D2, Adrenergic α1/α2, Histamine Receptor Antagonism
- Low-Moderate Serotonin 5-HT1C/5-HT1D/5-HT1A Receptor Antagonism
- Weak Dopamine D1 Receptor Antagonism
Selective α2-Adrenergic Receptor Antagonists
- Atipamezole (Antisedan)
- Idazoxan
- Mirtazapine (Remeron) (see Mirtazapine)
- Yohimbine (Actibine, Erex, Testomar, Yocon, Yohimar, Yohimbe) (see Yohimbine)
References
